Inhibitors

Lifitegrast /(3R,4R)-1-Benzyl-N,4-Dimethylpiperidin-3-Amine /顺式1-苄基-4- 甲基-3- 甲氨基-哌啶盐酸盐 /(2R,3R)-2,3-双[(4- 甲基苯甲酰基)氧基]丁二酸和 (3R,4R)-N,4-二甲基- 1-(苯基甲基)-3-哌啶胺的化合物 /4-Chloro-7-Tosyl-7H-Pyrrolo[2,3-D]Pyrimidine /4-Chloropyrrolo[2,3-D]Pyrimidine /2,4-Dichloro-7H-Pyrrolo (2,3-D)Pyrimidine /Oxymetholone /2-[ 1-(乙基磺酰基)-3-氮杂环丁亚基]乙腈 /(3R,4S)-3-(2-溴乙酰基)-4-乙基- 1-吡咯烷羧酸苄酯 /Cyclopropanecarboxylic acid (5-Bromo-[1,2,4]Triazolo[1,5-a]Pyridin-2-yl)-Amide /4-(Bromomethyl)Benzeneboronic Acid Pinacol Ester /4-[4-(4,4,5,5-四甲基[1,3,2]二氧硼杂环戊烷-2-基)苄基]硫代吗啉 1,1-二氧化物 /Carbamic acid,N-[5-[(4-Methylphenyl)Sulfonyl]-5H-Pyrrolo[2,3-b]Pyrazin-2-yl]-, Ethyl este /菲格替尼 /3-Cyclopentylacrylonitrile /(2S,5R)-5-Amino-2-Methylpiperidine-1-Carboxylic acid Benzyl Ester Hydrochloride /Pemigatinib /Ethyl (2S,3As,7As)-2,3,3A,4,5,6,7,7A-Octahydro-1H-Indole-2-Carboxylate,Hydrochloride /S-吲哚林-2-甲酸 /N-[(S)-乙氧羰基- 1-丁基]-(S)-丙氨酸 /2-(2-Butyl-4-Hydroxy-6-Methylpyrimidin-5-yl)-N,N-Dimethylacetamide /2-丁基- 1,6-二氢-N,N,4-三甲基-6-氧代- 1-[[2'-[ 1-(三苯甲基)- 1H-四氮唑-5-基][1, 1'-联苯]-4-基]甲基]-5-嘧啶乙酰胺 /2-[2-Butyl-4-Methyl-6-Oxo-1-[[4-[2-(2H-Tetrazol-5-Yl)Phenyl]Phenyl]Methyl]Pyrimidin-5-Yl]-N,N-Dimethylethanethioamide /(R)-叔丁基 (1-([1, 1'-联苯]-4-基)-3-羟基丙烷-2-基)氨基甲酸酯 /(R,E)-5-([1,1'-Biphenyl]-4-yl)-4-((tert-Butoxycarbonyl)Amino)-2-Methylpent-2-Enoic acid /(2R,4S)-5-(联苯-4-基)-4-[(叔丁氧基羰基)氨基]-2- 甲基戊酸 /N'-((2S,3S)-2-(Benzyloxy)Pentan-3-yl)Formohydrazide Oxalate /[(2S,3S)-2-(Benzyloxy)Pentan-3-yl]Hydrazine /(5R-cis)- 甲苯-4-磺酸 5-(2,4-二氟苯基)-5-( 1H- 1,2,4-三氮唑- 1-基)甲基四氢呋喃-3-基甲基酯 /2-[(1S,2S)- 1-乙基-2-苄氧基丙基]-2,4-二氢-4-[4-[4-(4-羟基苯基)- 1-哌嗪基]苯基]-3H- 1,2,4-三氮唑-3-酮 /Phenyl N-[4-[4-(4-Hydroxyphenyl)Piperazin-1-Yl]Phenyl]Carbamate /5-(2,4-二氟苯基)-5-(1,2,4-三唑-1-甲基)四氢呋喃-3-甲基]对氯苯磺酸酯 /4-(2-Bromoacetyl)Benzonitrile /2-甲胺基-3-吡啶甲;2-(甲氨基)-3-(羟甲基)吡啶 /(2-(((1-Chloroethoxy)Carbonyl)(Methyl)Amino)Pyridin-3-yl)Methyl 2-((tert-Butoxycarbonyl)(Methyl)Amino)Acetate /(2-(甲基氨基)吡啶-3-基)甲基 2-((叔丁氧羰基)(甲基)氨基)乙酸酯 /1-[[(2R,3S)-2-(2,5-二氟苯基)-3-甲基环氧乙烷基]甲基]-1H-1,2,4-三唑 /(2R,3R)-3-(2,5-Difluorophenyl)-3-Hydroxy-2-Methyl-4-(1H-1,2,4-Triazol-1-yl)Butanethioamide /1-[(2R,3R)-2-(2,4-Difluorophenyl)-2,3-Dihydroxybutyl]-1H-[1,2,4]Triazole Methanesulfonate Salt /4-Methylenepiperidine Hydrochloride /Cis-2,6-Dimethylmorpholine /2,4-二氯-3- 甲基苯甲酸 /(S)-(-)-3-(N-Methylamino)-1-(2-Thienyl)-1-Propanol /8-Bromooctanoic Acid /8-Bromooctanoic Acid Ethyl Ester /Carsalam /7-Hydroxy-1H-Quinolin-2-One /8-(2-羟基苯甲酰胺基)辛酸钠/SNAC /11-Chloro-2,3-Dihydro-2-Methyl-1H-Dibenz[2,3:6,7]Oxepino[4,5-C]Pyrrol-1-One /Trans-(+/-)-11-Chloro-2,3,3a,12b-Tetrahydro-2-Methyl-1H-Dibenz[2,3:6,7]Oxepino[4,5-c]Pyrrol-1-one /3-Nitro-4-((Tetrahydro-2H-Pyran-4-yl)Methylamino)Benzenesulfonamide /1H-Pyrrolo[2,3-B]Pyridin-5-Ol /1-((4'-氯-5,5-二甲基-3,4,5,6-四氢-[1,1'-联苯]-2-基)甲基)哌嗪 /1-[[2-(4-Chlorophenyl)-4,4-Dimethyl-1-Cyclohexen-1-yl]Methyl]Piperazine Dihydrochloride /2-((1H-吡咯并[2,3-b]吡啶-5-基)氧基)-4-溴苯甲酸叔丁酯 /2-Isopropyl-4-Methylpyridin-3-Amine /4-氯代苯并噻吩 /7-Chloro-6-Fluoro-1-(2-Isopropyl-4-Methylpyridin-3-yl)Pyrido[2,3-d]Pyrimidine-2,4(1H,3H)-Dione /Sotorasib /2-(Pyridin-2-Yldisulfanyl)Pyridine###2,2'-Dithiodipyridine /N-Succinimidyl 3-(2-Pyridyldithio)Propionate /Pantethine /阿拉格列汀中间体/2-甲基-吡唑并[1,5-a]嘧啶-6-羧酸 /N-(2-Amino-2-Methylpropyl)-2-Methylpyrazolo[1,5-a]Pyrimidine-6-Carboxamide /Ethyl 7-Chloro-8-Cyano-1-Cyclopropyl-6-Fluoro-4-oxo-1,4-Dihydroquinoline-3-Carboxylate /2-Chloro-3-Methyl-5-Bromopyridine /L-Homophenylalanine /L-Homophenylalanine Ethyl Ester Hydrochloride /维贝格龙中间体/Vibegron中间体 /3-Amino-4-Pyrazolecarbonitrile /4-氨基吡唑并[34-d]嘧啶 /3-Bromo-1H-Pyrazolo[3,4-d]Pyrimidin-4-Amine /3-Iodo-1H-Pyrazolo[3,4-D]Pyrimidin-4-Amine /(S)-1-Boc-3-Hydroxypiperidine /4-Amino-2-Methylpyrimidine-5-Carbonitrile /4-Amino-5-Aminomethyl-2-Methylpyrimidine, Dihydrochloride /3-(4-Phenoxyphenyl)-1H-Pyrazolo[3,4-d]Pyrimidin-4-Amine /2-(Hydroxy(4-Phenoxyphenyl)Methylene)Malononitrile /2-[Methoxy(4-Phenoxyphenyl)Methylene]Propanedinitrile /3-氨基-4-氰基-5-(4-苯氧基苯基)吡唑 /2-[2-(2-Fluorophenyl)-2-Oxoethyl]Propanedinitrile /5-(2-Fluorophenyl)-1H-Pyrrole-3-Carbonitrile /5-(2-Fluorophenyl)-1H-Pyrrole-3-Carbaldehyde /Pyridine-3-Sulfonyl Chloride /Oseltamivir Intermediate /Oseltamivir Phosphate /Phospho(Enol)Pyruvic Acid Monopotassium Salt###Phosphoenolpyruvic Acid Monopotassium Salt /3-Bromophenylhydrazine Hydrochloride /2-溴-1-氟-3-硝基苯 /3-(Dimethylamino)-2-Fluoro-1-(4-Methyl-2-(Methylamino)-Thiazol-5-yl)prop-2-en-1-one /6,7,8-Trifluoro-1-(Formylmethylamino)-1,4-Dihydro-4-oxo-3-Quinolinecarboxylic acid Ethyl Ester /(R)-3-Chloro-4-(2,3-Dihydroxypropoxy)Benzaldehyde /(Z) -2- (Propylimino) -3- (o-Methylphenyl) Thiazolidine-4-one /2-Bromo-4-Fluoronitrobenzene /2-Ethyl-4-Fluoro-1-Nitrobenzene /(3,3-Difluoro-1-Methyl-Cyclobutyl)Methanol /2,2',3,3'-Tetrahydro-1,1'-Spirobi[1H-Indene]-7,7'-Diol /(1S,5R)-Ethyl 2-oxo-3-Oxabicyclo[3.1.0]Hexane-1-Carboxylate /4-Hydroxy-5-Methyl-1H-Pyridin-2-one /1,1,1-Trifluoro-3-Iodobutane /Benzoic acid, 3,4-Dihydroxy-2-Methyl-, Methyl Ester /1,3,5-Trisilacyclohexane /5-Formyl-4-Methyl-1H-Indole-2-Carbonitrile /5-Vinylpyrrolidone /3,5,6-Trichloro-1,2,4-Triazine /2-((tert-Butyldimethylsilyl)oxy)Ethane-1-Sulfonyl Chloride /氯乙基吗啉盐酸盐(特班布林中间体）/N-(2-氯乙基)吗啉盐酸盐 /1-(2-Chloroethyl)Piperidine,Hydrochloride /Ethyl 2-Oxocyclohexanecarboxylate /1-Boc-3-Hydroxypiperidine /6-Chloro-2-Methyl-2H-Indazol-5-Amine /3-(tert-Butyl)-6-(Ethylthio)-1,3,5-Triazine-2,4(1H,3H)-Dione /Ensitrelvir /异丁酰胺基噻唑基间苯二酚 /叔丁基(S)-(1-(3-溴-6-(3-甲基-3-(甲基磺酰基)- 1-炔-1-基)吡啶-2-基)-2-(3,5-二氟苯基)乙基)氨基甲酸酯 /4-氯-7-(4,4,5,5-四甲基-1,3,2-二氧杂硼烷-2-基)-1-(2,2,2-三氟乙基)-1H-吲唑-3-胺 /2-((3bS,4aR)-5,5-二氟-3-(三氟甲基)-3b,4,4a,5-四氢-1H-环丙烯并[3,4]环戊二烯并[1,2-c]吡唑-1-基)乙酸 /3-甲基-3-(甲基磺酰基)-1-丁炔;3-甲基-3-(甲基磺酰基)丁-1-炔 /(R）-4-甲基-1，3，2-二恶噻戊环2，2-二氧化物 /5-Bromoindole-2-Carboxylic Acid /(S)-5-(2,2-二甲基四氢-2H-吡喃-4-基)-N-甲基-N-苯基-1H-吲哚-2-甲酰胺 /4-氟-3,5-二甲基苯基肼盐酸盐 /5-溴-4-氟-1-甲基-1H-吲唑 /(S)-2-(4-氟-3,5-二甲基苯基)-4-甲基-3-(2-氧代-2,3-二氢-1H-咪唑-1-基)-2,4,6,7-四氢-5H-吡唑并[4,3-C]吡啶-5-羧酸叔丁酯 /5-((S)-2,2-Dimethyltetrahydro-2H-Pyran-4-yl)-1-((1S,2S)-2-Methyl-1-(5-oxo-4,5-Dihydro-1,2,4-Oxadiazol-3-yl)Cyclopropyl)-1H-Indole-2-Carboxylic acid /(4AS,8AS,9S)-9-(二甲基氨基)-4A-[[叔丁基二甲基硅烷基]氧基]-8A,9-二氢-3-(苯基甲氧基)-萘并[2,3-D]异恶唑-4,5(4AH,8H)-二酮 /tert-butyl (S)-5-cyano-4-hydroxy-6-methyl-3,6-dihydropyridine-1(2H)-carboxylate /2-(苄氧基)-3-(苄基氨基)-5-氟-6-甲基苯甲酸 /3-甲氧基-2-呋喃醛 /2-(1-吡咯烷基)乙酸盐酸盐 /(S)-1-(3-(苄氧基)异恶唑-5-基)-N,N-二甲基丙-2-烯-1-胺 3-羧基-2,3-二羟基丙酸酯 /3-(3-氯-1,2,5-噻二唑-4-基)-吡啶 /3-(4-己氧基-1,2,5-噻二唑-3-基)-1-甲基吡啶碘化物 /Silane, (1,1-Dimethylethyl)Dimethyl[[(3β,5E,7E)-9,10-Secocholesta-5,7,10(19)-Trien-3-yl]oxy]- /阿尔法骨化醇双TBS中间体/((1R,3S,E)-5-((E)-2-((1R,3aS,7aR)-7a-methyl-1-((R)-6-methylheptan-2-yl)dihydro-1H-inden-4(2H,5H,6H,7H,7aH)-ylidene)ethylidene)-4-methylenecyclohexane-1,3-diyl)bis(oxy)bis(tert-butyldimethylsilane) /阿法骨化醇中间体 /(1Α,3Β,5E,7E)-20-羟甲基-9,10-开环胆甾-1,3,-双叔丁基二甲基硅氧基-5,7,10(19)-三烯 /艾地骨化醇中间体 /24-羰基-1,3-双TBS-反式-钙泊三醇 /双(叔丁基二甲基硅基)-反式-钙泊三醇/G10 /Calcipotriol###Calcipotriene /Calcipotriol Monohydrate /(7Ar)-1-(6-羟基-5,6-二甲基庚-3-烯-2-基)-7a-甲基-1,2,3,3a,4,5,6,7-八氢茚-4-醇 /帕里骨化醇A环 /Paricalcitol###Paricalcitol /骨化三醇N-3 /5,6-Trans-1Alpha,25-Dihydroxyvitamin D3 /Calcitriol /(Z)-2-((3S,5R)-3,5-双((叔丁基二甲基硅基)氧代)-2-甲烯基亚环己基)乙基-1-醇 /骨化三醇双TBS /A环双TBS中间体 /氟骨化醇 /(ε r,1R,3aR,4S,7aR)-八氢-4-羟基-ε,7a-二甲基-α,α-二(三氟甲基)-1H-茚- 1-戊醇 /(1R,3S,5Z)-5-[(2E)-2-[(1R,3As,7Ar)-1-[(2R,5R)-5-Hydroxy-6-Methylheptan-2-Yl]-7A-Methyl-2,3,3A,5,6,7-Hexahydro-1H-Inden-4-Ylidene]Ethylidene]-4-Methylidenecyclohexane-1,3-Diol /他骨化醇一水物 /(2Z)-2-[(3R,4R,5R)-3,5-双[[(1,1-二甲基乙基)二甲基甲硅烷基]氧基]-4-[3-[[(1,1-二甲基乙基)二甲基甲硅烷基]氧基]丙氧基]-2-亚甲基环己基]乙基]二苯基-氧化膦 /(Z)-[2-{(3R,4R,5R)-3,5-双(叔丁基二甲基硅烷氧基)-2-亚甲基-4-(3-(叔丁基二苯基硅烷氧基)丙氧基)亚环己基}乙基]二苯基氧化膦 /(1R,3aR,4S,7aR)-1-[(2R)-6-羟基-6- 甲基庚-2-基]-7a-甲基八氢-1H-茚-4-醇 /艾地骨化醇N-1 /Eldecalcitol /25-羟基维生素D2, 25-羟麦角甾醇 /1α ,25-二羟基维生素D2 /Maxacalcitol /骨化二醇一水合物;25-羟基维生素D3一水合物 /依奈骨化醇;伊奈骨化醇 /Calcidiol /Eb 1089,(1R,3S,5Z)-5-[(2E)-2-[(1R,3As,7Ar)-1-[(1R,2E,4E)-6-Ethyl-6-Hydroxy-1-Methyl-2,4-Octadien-1-Yl]-Octahydro-7α-Methyl-4H-Inden-4-Ylidene]Ethylidene]-4-Methylene-1,3-Cyclohexanediol /来沙骨化醇 /阿托骨化醇 /CD二醇 /CD二醇单TBS /G6侧链;1-环丙基-2-(三苯基膦亚基)乙酮 /Tert-Butyl-[3-(2-Diphenylphosphorylethylidene)-4-Methylidenecyclohexyl]Oxy-Dimethylsilane /帕夫骨化醇 /5-((R)-2-((1R,3aS,7aR,E)-4-((Z)-2-((3S,5R)-3,5-dihydroxy-2-methylenecyclohexylidene)ethylidene)-7a-methyloctahydro-1H-inden-1-yl)propyl)-3-methylenedihydrofuran-2(3H)-one /TEI-9647 /(3aR,4R,5R,6aS)-5-(tert-butyldimethylsilyloxy)-4-((R)-3-(tert-butyldimethylsilyloxy)-5-phenylpentyl)hexahydro-2H-cyclopenta[b]furan-2-one /Latanoprost /Travoprost /[1,1'-Biphenyl]-4-carboxylic acid, (3aR,4R,5R,6aS)-4-[(1E)-3,3-difluoro-4-phenoxy-1-buten-1-yl]hexahydro-2-oxo-2H-cyclopenta[b]furan-5-yl ester /他氟前列腺素 /(E)-7-[(1R,2R,3R)-3-Hydroxy-2-[(E,3S,5S)-3-Hydroxy-5-Methylnon-1-Enyl]-5-Oxocyclopentyl]Hept-2-Enoic Acid###Limaprost /Triphenyl(3-Phenylmethoxypropyl)Phosphanium,Bromide /[(4S)-4-Methyl-2-oxooctyl]phosphonic acid dimethyl ester /Lubiprostone /贝美前列腺素 /Prostaglandin E1 /Vitamin D2 /Alfacalcidol /Tofacitinib Citrate /托吡司特 /Upadacitinib /Iguratimod /伏诺拉生 /2-[(4-Methoxy-3-Methylpyridin-2-Yl)Methylsulfinyl]-6-Pyrrol-1-Yl-1H-Benzimidazole /Mirogabalin Besylate /Florfenicol /布瑞哌唑 /Disodium,[2,6-Di(Propan-2-Yl)Phenoxy]Methyl Phosphate /Deoxycholic Acid###Deoxycholic Acid /Pranoprofen /雷芬那辛 /Tulobuterol /Bepotastine Besylate###Bepotastine Besilate /Emedastine Difumarate###Emedastine Fumarate /Sodium,4-[2-Hydroxy-1-[(E)-3-Hydroxy-4-Methyloct-1-En-6-Ynyl]-2,3,3A,8B-Tetrahydro-1H-Cyclopenta[B][1]Benzofuran-5-Yl]Butanoate###Beraprost Sodium /Sacubitril Valsartan /非马沙坦钾三水合物 /Selexipag /Isavuconazole /Efinaconazole /8-（2-羟基苯甲酰胺基）辛酸钠 /10-(2-羟基苯甲酰胺基)奎酸钠 /8-(4-氯-2-羟基苯甲酰氨基)辛酸钠 /N-(5-氯-2-羟基苯甲酰)-8-氨基辛酸 /8-(2-羟基苯甲酰氨基)辛酸精氨酸盐 /精氨酸正葵酸盐 /精氨酸正辛酸盐 /赖氨酸正葵酸盐 /Lysine Caprylate /Lauroyl-L-Carnitine Chloride /6,6'-Dibehenoyl-Alpha,Alpha'-Trehalose